PHTHALAZINE KETONE DERIVATIVE, METHOD OF OBTAINING THEREOF AND PHARMACEUTICAL APPLICATION Russian patent published in 2015 - IPC C07D487/04 A61K31/502 A61P35/00 

Abstract RU 2564527 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to a phthalazine ketone derivative, represented by formula in which radicals and symbols have values, given in the invention formula, a method of its obtaining, a pharmaceutical composition, containing the claimed derivative, and its application as a poly(ADP-ribose)polymerase (PARP) inhibitor.

EFFECT: obtaining the pharmaceutical composition for application as the poly(ADP-ribose)polymerase (PARP) inhibitor.

13 cl, 26 ex

Similar patents RU2564527C2

Title Year Author Number
BICYCLIC LACTAMS AND METHODS FOR USE THEREOF 2016
  • Patel Snakhel
  • Gamilton Gregori
  • Stivala Krejg
  • Chen Khuejfen
  • Chzhao Gujlin
RU2716136C2
IMIDAZOPYRAZINE OR IMIDAZODIAZEPINE DERIVATIVES, ACTIVE WITH RESPECT TO RECEPTOR CB2 2008
  • Betskett R. Paul
  • Foster Richard
  • Khenault Christelle
  • Ralbovsky Dzhanet L
  • Gauss Karla M
  • Gustafson Gari R
  • Luo Zhijong
  • Kampbell Anna-Mari
  • Shelekkhin Tat'Jana E
RU2540074C2
HETEROCYCLIC COMPOUNDS AS PRMT5 INHIBITORS 2018
  • Vadivelu, Saravanan
  • Rajagopal, Sridharan
  • Burri, Raghunadha Reddy
  • Garapaty, Shivani
  • Sivanandhan, Dhanalakshmi
  • Thakur, Manish Kumar
  • Natarajan, Tamizharasan
  • Swamy, Indu N
  • Nagaraju, Nagendra
  • Kanagaraj, Subramaniam
  • Mohd, Zainuddin
  • Sarkar, Sayantani
  • Samanta, Swapan Kumar
  • Hariprakash
RU2797822C2
TETRAHYDRO-IMIDAZO[1,5-A]PYRAZINE DERIVATIVE SALTS, METHODS FOR PREPARING THEM AND MEDICAL APPLICATION THEREOF 2010
  • Tan Pehn Cho
  • Sun' Pjaojan
  • Jan Fanlon
  • Ljan Tszin'Dun
  • Shehn' Guanjuan'
  • Van Jan
  • Fan' Tszjan
RU2523543C2
COMPOUND BASED ON DIHYDRONAPTHYRIDINONE, METHOD OF ITS OBTAINING, AND ITS USE IN MEDICINE 2021
  • Zhou, Fusheng
  • Xu, Xiaoming
  • Zhang, Leitao
  • Li, Xin
  • Tang, Lili
  • Lan, Jiong
RU2809869C1
PYRROLOPYRAZINE KINASE INHIBITORS 2012
  • Chen Shaotsin
  • De Visente Fidalgo Khaver
  • Gamilton Metyu Majkl
  • Germann Jokhannes Kornelius
  • Kennedi-Smit Dzhoshua
  • Li Khuntszyuj
  • Lavi Allen Dzhon
  • Lukas Metyu S.
  • Lyuk Kin-Chun Tomas
  • Linch Stiven M.
  • O'Yang Kaund
  • Pedilla Fernando
  • Shoenfeld Rajan Krejg
  • Sidduri Achyutarao
  • Sot Majkl
  • Van Tse
  • Vovkulich Piter Majkl
  • Chzhan Syaokhu
RU2673064C2
BICYCLIC 6-ALKYLIDENEPENEMS AS β-LACTAMASE INHIBITORS 2003
  • Venkatesan Aranapakam Mudumbaj
  • Mansour Tarek Sukhajl
  • Abe Takao
  • Jamamura Itsuki
  • Takasaki Tsujosi
  • Agarval Atul
  • Santos Osval'Do Dos
  • Sum Fuk-Vakh
  • Lin Jang-I
RU2339640C2
BICYCLIC HETEROCYCLIC COMPOUNDS AND THEIR APPLICATIONS 2020
  • Kregg, Dzhejms Dzhozef
  • Bakl, Andreas
  • Aaj, Naing
  • Tambo-Ong, Arlin A.
  • Koltun, Elena S.
  • Dzhill, Edrian Liam
  • Tompson, Severin
  • Glidt, Mika Dzh.
RU2811612C2
EP4 ANTAGONISTS 2016
  • Zheng Wanjun
  • Zhu Xiaojie
  • Du Hong
  • Postema Maarten
  • Jiang Yimin
  • Li Jing
  • Yu Robert
  • Choi Hyeong-Wook
  • Lee Jaemoon
  • Fang Frank
  • Custar Daniel
RU2761341C2
CLASS OF BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUNDS FOR TARGETED DESTRUCTION OF ANDROGEN RECEPTORS AND USE THEREOF 2020
  • Du, Vu
  • Ven, Kun
  • Fu, Ivej
  • Lv, Khajbin
  • Khe, Tszinyun
  • Tsin, Dekun
  • Li, Yuj
  • Duan, Tszini
  • Li, Yun
  • Aj, Chaovu
  • Tu, Chzhilin
  • Chen, Yuanvej
  • Li, Sinkhaj
  • Li, Khajbo
RU2825000C2

RU 2 564 527 C2

Authors

Tan Pehn Cho

Li Sin'

Li Sjantsin'

Chehn' Jan

Van Bin'

Chzhu Chzhe

Dates

2015-10-10Published

2011-07-26Filed