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2 579 515

(13)

(51)

IPC

C07D231/38(2006-01-01)

A61K31/415(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2014154122/04, 2014-12-29

(24)

Start date

2014-12-29

(22)

Actual filing date

2014-12-29

(45)

Published

2016-04-10

(72)

Inventor

Ljubjashkin Aleksej ViktorovichKomar Natalja AndreevnaSuboch Georgij AnatolevichTovbis Mikhail SemenovichPerjanova Olga Vladimirovna

(73)

Holder

Federalnoe Gosudarstvennoe Bjudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovanija Gosudarstvennyj Tekhnologicheskij Universitet"

ALKOXYMETHYL-SUBSTITUTED 1H-4-AMINOPYRAZOLES Russian patent published in 2016 - IPC C07D231/38 A61K31/415 A61P31/04

Abstract RU 2579515 C1

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to new alkoxymethyl-substituted 1H-4-aminopyrazoles having the following formula, with the phenyl (C₆H₅), or naphthyl (C₁₀H₇) substitute having antibacterial activity. These substances have high bactericidal and bacteriostatic activity.

EFFECT: detected properties of substances obtained make it possible to apply them in pharmacology for creation of antibacterial preparations.

1 cl, 2 ex

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RU 2 579 515 C1

Authors

Ljubjashkin Aleksej Viktorovich

Komar Natalja Andreevna

Suboch Georgij Anatolevich

Tovbis Mikhail Semenovich

Perjanova Olga Vladimirovna

Dates

2016-04-10—Published

2014-12-29—Filed