OBTAINING INTERMEDIATE PRODUCTS FOR SYNTHESIS OF POSACONAZOLE Russian patent published in 2016 - IPC C07D405/06 C07D405/14 

Abstract RU 2580318 C2

FIELD: chemistry.

SUBSTANCE: claimed invention relates to method for obtaining chiral compound of formula or its salt, where Y1 and Y2 independently stand for F or Cl, preferably F, as well as to crystalline chiral compound of formula (IX) or its salt, in which from 80 to 95%, preferably from 85 to 95% of molecules of said crystalline compound or its salt are contained in form of cis-isomer of formula or its salt and from 20 to 5%, preferably from 15 to 5% of molecules of said crystalline compound or its salt are contained in form of trans-isomer of formula or its salt, and to its application for obtaining fungicidal preparation.

EFFECT: increase of method efficiency.

23 cl, 5 dwg, 2 tbl, 2 ex

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RU 2 580 318 C2

Authors

De-Suza Dominik

Joshi Shrirang V.

Bkhuta Zachin

Pajz Abkhinaj S.

Chavan Dattatraja N.

Metkar Shashikant D.

Dates

2016-04-10Published

2011-05-18Filed