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2 584 653

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IPC

A61K38/05(2006-01-01)

A61K9/22(2006-01-01)

A61P25/18(2006-01-01)

(21) (22)

Application

2012135595/15, 2012-08-20

(24)

Start date

2012-08-20

(22)

Actual filing date

2012-08-20

(45)

Published

2016-05-20

(72)

Inventor

Seredenin Sergej BorisovichPjatin Boris MikhajlovichAvdjunina Nina IvanovnaAlekseev Konstantin ViktorovichGrushevskaja Ljubov NikolaevnaBlynskaja Evgenija ViktorovnaTikhonova Natalja ViktorovnaGaevaja Ljudmila MikhajlovnaUstinova Marija IsaakovnaOstrovskaja Rita UsherovnaSergeeva Marija Sergeevna

(73)

Holder

Federalnoe Gosudarstvennoe Bjudzhetnoe Nauchnoe Uchrezhdenie Institut Farmakologii Imeni V.V. Zakusova"

PHARMACEUTICAL COMPOSITION WITH PROLONGED RELEASE WITH ANTIPSYCHOTIC ACTIVITY AND SYNTHESIS METHODS THEREOF Russian patent published in 2016 - IPC A61K38/05 A61K9/22 A61P25/18

Abstract RU 2584653 C2

FIELD: pharmaceutics.

SUBSTANCE: group of inventions refers to pharmacy and medicine and concerns prolonged pharmaceutical composition possessing antipsychotic action and containing as medicinal substance therapeutically effective amount of methyl ether of N-caproil-L-prolyl-L-tyrosine and, as auxiliary substances-prolonging polymers, filler, anti-friction substance, film casing. Invention also discloses methods for preparing said composition (versions).

EFFECT: group of inventions provides prolonged release of active substance, as well as allows to reduce rate of application, reducing vibrations of active substance concentration in blood.

31 cl, 13 ex, 7 tbl

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RU 2 584 653 C2

Authors

Seredenin Sergej Borisovich

Pjatin Boris Mikhajlovich

Avdjunina Nina Ivanovna

Alekseev Konstantin Viktorovich

Grushevskaja Ljubov Nikolaevna

Blynskaja Evgenija Viktorovna

Tikhonova Natalja Viktorovna

Gaevaja Ljudmila Mikhajlovna

Ustinova Marija Isaakovna

Ostrovskaja Rita Usherovna

Sergeeva Marija Sergeevna

Dates

2016-05-20—Published

2012-08-20—Filed