COMPOUNDS HAVING ANTAGONISTIC ACTIVITY TOWARDS MUSCARINIC RECEPTORS AND AGONIST ACTIVITY TO BETA2-ADRENORECEPTORS Russian patent published in 2017 - IPC C07D401/12 C07D409/14 C07D413/12 C07D417/12 A61K31/4545 A61K31/4709 A61P11/06 A61P11/08 

Abstract RU 2606121 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to compounds of general formula (I),

acting as muscarinic receptors antagonists or beta2-adrenoreceptors agonists, as well as to pharmaceutical compositions based thereon and to therapeutic applications for preparing a medicine to prevent and treat diseases, such as asthma, chronic bronchitis, etc.

EFFECT: obtained are novel compounds of formula (I) having activity towards muscarinic receptors or beta2-adrenoreceptors.

13 cl, 5 tbl, 39 ex, 2 dwg

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RU 2 606 121 C2

Authors

Rankati Fabio

Linnej Jen

Ritstsi Andrea

Blekebi Uesli

Najt Kris

Dates

2017-01-10Published

2012-06-07Filed