FIELD: chemistry.
SUBSTANCE: invention relates to compounds of formula I
wherein R1 is selected from the group consisting of formula 
(1), formula 
(2),
formula 
(3), for the manufacture and delivery of conjugated molecules, such as small molecules, peptides, nucleic acids, fluorescent molecules and polymers that are associated with the integrin antagonists of VLA-4, target cells expressing VLA-4.
EFFECT: improved properties of compounds.
16 cl, 6 dwg, 5 tbl, 14 ex
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