FIELD: chemistry.
SUBSTANCE: invention relates to compounds of formula
wherein R1 is selected from compounds
(1) 
(2) 
(3), which are used for the manufacture and delivery of conjugated groups, such as small molecules, peptides, nucleic acids, fluorescent groups and polymers crosslinked with antagonists of integrin LFA-1 for targeted delivery to cells expressing LFA-1.
EFFECT: improved properties.
21 cl, 6 dwg, 1 tbl, 10 ex
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