TRPV1 ANTAGONISTS AND USE THEREOF Russian patent published in 2012 - IPC C07D401/04 C07D401/14 C07D417/12 C07D417/14 A61K31/4545 A61P23/00 

Abstract RU 2452733 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of formula 1 or pharmaceutically acceptable derivatives thereof, where values of radicals X, W, R4, Ar1, Ar2, R3, R4, R20 are as described in paragraph 1 of the claim. The invention also describes a composition for treating or preventing pain, UI, ulcers, inflammatory bowel disease or irritable bowel syndrome.

EFFECT: compound which can be used in medicine is obtained and described.

46 cl, 10 ex, 1 tbl

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RU 2 452 733 C2

Authors

Tafess Lehjkea

Kurose Norijuki

Dates

2012-06-10Published

2008-04-25Filed