PROCESS FOR PREPARATION OF 4-[5-(PYRIDIN-4-YL)-1H-1,2,4-TRIAZOL-3-YL]PYRIDINE-2-CARBONITRILE AND ITS INTERMEDIATE Russian patent published in 2018 - IPC C07D213/86 

Abstract RU 2644766 C2

FIELD: pharmaceutics.

SUBSTANCE: invention relates to compound of formula (4) and industrially useful process for preparation of pharmaceutically valuable 4-[5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl]pyridine-2-carbonitrile (1) and intermediate (4) to obtain this compound. Process for preparing compound is represented by the following reaction scheme: .

EFFECT: industrially useful process for preparation of pharmaceutically valuable 4-[5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl]pyridine-2-carbonitrile.

4 cl, 3 ex

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RU 2 644 766 C2

Authors

Ivabuti Josiyuki

Miyata Satikho

Uda Dzunitiro

Nagata Osamu

Dates

2018-02-14Published

2013-07-24Filed