1-(SUBSTITUTED BENZOYL)-5-FLUORO-4-IMINO-3-METHYL-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE DERIVATIVES Russian patent published in 2018 - IPC C07D239/47 A01N43/54 A01P3/00 

Abstract RU 2656101 C2

FIELD: crop growing.

SUBSTANCE: present invention relates to a compound of formula (I) or a salt thereof, or a hydrate thereof. Such a fungal disease is a fungal disease selected from the group consisting of Venturia inaequalis, Septoria tritici, Cercospora beticola, Cercospora arachidicola, Cercosporidium personatumI and Mycosphaerella fijiensis, mainly Septoria tritici. In the compound of formula (I)

is -C(=O)R4; R2 is C1-C6alkyl; R3 is H; R4 is phenyl, which may be optionally substituted with 1 to 3 R5 groups; and R5 is independently halogen or C1-C6alkyl. Preferred salts of the compound are its hydrochloride, hydrobromide or hydroiodide. Invention also relates to a composition for controlling fungal diseases of plants using said compound, which can be made in a form suitable for application to the soil, plant, part of the plant, leaf and/or plant seed, and to a method of combating fungal infection or preventing fungal infection of plants. Fungicidally effective amount of at least one of said compounds is applied to at least one surface, selected from the part of the plant, the area near the plant, the soil in contact with the plant, the soil near the plant, any surface near the plant, any surface in contact with the plant, seeds and equipment used in the cultivation of plants.

EFFECT: compounds have fungicidal activity and can be used to control or prevent fungal diseases of plants.

19 cl, 2 ex, 3 tbl

Формула (I) - Formula (I)

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RU 2 656 101 C2

Authors

Lorsbakh Bet

Ouen U. Dzhon

Yao Chenlin

Stelzer Lindsej

Dates

2018-05-31Published

2013-12-23Filed