CRYSTALLINE ALLISARTAN ISOPROXIL, METHOD FOR PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITION Russian patent published in 2018 - IPC C07D403/10 A61K31/4178 A61P9/12 

Abstract RU 2662816 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a crystalline form of allisartan isoproxil which has diffraction peaks at diffraction angles (2θ±0.2°) 6.9, 8.0, 13.8, 20.1, 21.1, 22.2, 24.0 and 27.7 in spectra of pRSA. Invention also relates to a pharmaceutical composition of allisartan isoproxil for the treatment of hypertensive diseases.

EFFECT: produced is a novel crystalline form of allisartan isoproxil, having good mobility and high stability.

11 cl, 7 dwg, 8 ex

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RU 2 662 816 C2

Authors

Tan Duanmin

Ou Tszyun

Dates

2018-07-31Published

2015-06-05Filed