DNA-PK INHIBITORS Russian patent published in 2018 - IPC C07D413/02 A61K31/517 A61K31/5377 A61P35/00 

Abstract RU 2676259 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to new compounds of formula (I), to pharmaceutically acceptable compositions containing these compounds and to methods for using the compositions for treating cancer. (I).

EFFECT: obtained new compounds suitable to be used as inhibitors of DNA-PK.

64 cl, 2 tbl, 7 ex

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RU 2 676 259 C2

Authors

Maksvell Dzhon Patrik

Charifson Pol S.

Tan Tsin

Ronkin Stiven M.

Dzhekson Katrina Li

Pirs Albert Charlz

Lauffer Devid Dzh.

Li Pan

Zhiru Simon

Syuj Tszinvan

Kottrell Kevin M.

Morris Mark A.

Vaal Natan D.

Kort Dzhon Dzh.

Gu Vensin

Den Khunbo

Dates

2018-12-27Published

2014-03-12Filed