FIELD: chemistry.
SUBSTANCE: invention relates to a method of producing triazine, pyrimidine and pyridine derivatives of formula (I) by condensation of the corresponding halogen-triazine, pyrimidine or pyridine via a coupling reaction of Suzuki with pyridyl- or pyrimidinyl-borane, where the amino-functional group is protected in form of formamidine. Invention also relates to suitable intermediate compounds and methods of producing said intermediate compounds.
.
EFFECT: technical result is a novel method of producing compounds of formula (I), which enables to obtain desired compounds with high output and purity.
19 cl, 3 tbl, 17 ex, 1 dwg
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