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2 699 658

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IPC

C07D451/04(2006-01-01)

A61K31/46(2006-01-01)

A61P25/06(2006-01-01)

(21) (22)

Application

2016133999, 2016-08-19

(24)

Start date

2016-08-19

(22)

Actual filing date

2016-08-19

(45)

Published

2019-09-09

(72)

Inventor

Kostochka Leonid MikhajlovichGanshina Tamara SergeevnaNaplekova Polina LeonidovnaNarkevich Viktor BorisovichVoronina Tatyana AleksandrovnaKudrin Vladimir SergeevichMirzoyan Ruben SimonovichKurdyumov Ilya NikolaevichGudasheva Tatyana AleksandrovnaZherdev Vladimir PavlovichPyatin Boris MikhajlovichGorbunov Aleksandr Anatolevich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Nauchnoe Uchrezhdenie Institut Farmakologii Imeni V.V. Zakusova"

ACYLHYDRAZONE (2,3,4-TRIMETHOXY-N'-(8-METHYL-8-AZABICYCLO[3.2.1.]OCTANE-3-YLIDENE) BENZOHYDRAZIDE HYDROCHLORIDE), HAVING ANTIMIGRAINE AND ANXIOLYTIC ACTIVITY Russian patent published in 2019 - IPC C07D451/04 A61K31/46 A61P25/06

Abstract RU 2699658 C2

FIELD: chemistry.

SUBSTANCE: invention relates to acyl hydrazone (2,3,4-trimethoxy-N'-(8-methyl-8-azabicyclo[3.2.1.]octane-3-ylidene) benzohydrazide hydrochloride) of structural formula (I), which can be used in medicine:

EFFECT: disclosed is a new compound with antimigraine and anxiolytic activity.

1 cl, 3 ex, 3 tbl, 1 dwg

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RU 2 699 658 C2

Authors

Kostochka Leonid Mikhajlovich

Ganshina Tamara Sergeevna

Naplekova Polina Leonidovna

Narkevich Viktor Borisovich

Voronina Tatyana Aleksandrovna

Kudrin Vladimir Sergeevich

Mirzoyan Ruben Simonovich

Kurdyumov Ilya Nikolaevich

Gudasheva Tatyana Aleksandrovna

Zherdev Vladimir Pavlovich

Pyatin Boris Mikhajlovich

Gorbunov Aleksandr Anatolevich

Dates

2019-09-09—Published

2016-08-19—Filed