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2 803 750

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IPC

C07D211/58(2006-01-01)

A61K31/44(2006-01-01)

A61K31/4468(2006-01-01)

A61P25/06(2006-01-01)

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Application

2022133685, 2022-12-21

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Start date

2022-12-21

(22)

Actual filing date

2022-12-21

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Published

2023-09-19

(72)

Inventor

Ganshina Tamara SergeevnaKostochka Leonid MikhajlovichKurza Elena VladimirovnaKurdyumov Ilya NikolaevichMaslennikov Denis VadimovichGnezdilova Anna ViktorovnaMirzoyan Ruben SimonovichKovalev Georgij IvanovichVasileva Ekaterina ValerevnaAbdullina Aliya AnvyarovnaVakhitova Yuliya VenerovnaSeredenin Sergej Borisovich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Nauchnoe Uchrezhdenie Institut Farmakologii Imeni V.V. Zakusova"

COMPOUND OF 2,3,4-TRIMETHOXY-N-(2,2,6,6-TETRAMETHYLPIPERIDIN-4-YLIDENE)BENZOHYDRAZIDE HYDROCHLORIDE WITH ANTISEROTONIN CEREBROVASCULAR AND ANTIMIGRAINE ACTIVITY Russian patent published in 2023 - IPC C07D211/58 A61K31/44 A61K31/4468 A61P25/06

Abstract RU 2803750 C1

FIELD: pharmaceutical industry.

SUBSTANCE: invention relates to the compound 2,3,4-trimethoxy-N-(2,2,6,6-tetramethylpiperidin-4-ylidene)benzohydrazide hydrochloride.

EFFECT: connection as an antiserotonin cerebrovascular and anti-migraine agent, belongs to low-hazard substances (toxicity class 4), does not cause undesirable side effects, significantly exceeds tropane derivatives in terms of economic feasibility of synthesis.

1 cl, 11 tbl, 6 ex

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RU 2 803 750 C1

Authors

Ganshina Tamara Sergeevna

Kostochka Leonid Mikhajlovich

Kurza Elena Vladimirovna

Kurdyumov Ilya Nikolaevich

Maslennikov Denis Vadimovich

Gnezdilova Anna Viktorovna

Mirzoyan Ruben Simonovich

Kovalev Georgij Ivanovich

Vasileva Ekaterina Valerevna

Abdullina Aliya Anvyarovna

Vakhitova Yuliya Venerovna

Seredenin Sergej Borisovich

Dates

2023-09-19—Published

2022-12-21—Filed