THIENO[3,2-d]PYRIMIDINE DERIVATIVES WITH PROTEIN KINASE INHIBITORY ACTIVITY Russian patent published in 2019 - IPC C07D495/04 C07D215/02 

Abstract RU 2705577 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to a process for the preparation of thieno[3,2-d]pyrimidine compound of formula (I), or a pharmaceutically acceptable salt thereof, which comprises the steps of 1–3:

.

Invention also relates to a process for the preparation of a compound of formula

.

Radical values are given in claim 1.

EFFECT: method of preparing a pharmaceutically acceptable salt is provided.

17 cl, 125 ex, 5 tbl

Similar patents RU2705577C2

Title Year Author Number
TIENOPYRIMYDINE [3,2-D] PRODUCTION, WHICH HAS INHIBITORY ACTIVITY AGAINST PROTEIN KINASES 2012
  • Bae In Khvan
  • Son Dzung Beom
  • Khan Sang Mi
  • Kvak Eun Dzoo
  • Kim Kho Seok
  • Song Dzi Joung
  • Biun Eun Joung
  • Dzun Seung Akh
  • Akhn Joung Gil
  • Sukh Kvee Khiun
RU2625799C2
THIENO[3,2-d]PYRIMIDINE DERIVATIVES, POSSESSING INHIBITING ACTION WITH RESPECT TO PROTEINKINASE 2011
  • Son Dzung Beom
  • Dzung Seung Khiun
  • Choj Va Il
  • Dzung Joung Khee
  • Choj Dzae Jul
  • Song Dzi Jeon
  • Li Kiu Khang
  • Li Dzae Chul
  • Kim Eun Joung
  • Akhn Jung Gil
  • Kim Maeng Sup
  • Choj Khvan Geun
  • Sim Tae Bo
  • Kham Joung Dzin
  • Park Dong-Sik
  • Kim Khvan
  • Kim Dong-Vook
RU2524210C2
NEW AMINOARYL DERIVATIVE SUITABLE AS A DIACYLGLYCEROLACYL TRANSFERASE 2 INHIBITOR AND ITS APPLICATION 2020
  • Yoon, Seung Hyun
  • Joo, Hyun Woo
  • Seo, Bo Kyung
  • Lee, Eun Jin
  • Jung, Jin Young
  • Yoon, Su Young
  • Cho, Woo Young
RU2799819C1
NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHIBITION OF TYROSINE KINASE ACTIVITY 2011
  • Cha Mi Yang
  • Kang Seok Dzong
  • Kim Mi Ra
  • Li Dzu Jeon
  • Dzeon Dzi Yang
  • Dzo Mioung Gi
  • Kvak Eun Dzoo
  • Li Kvang Ok
  • Kha Tae Khee
  • Sukh Kvee Khiun
  • Kim Maeng Sup
RU2585177C2
BICYCLIC DIHYDROPYRIMIDINECARBOXAMIDE DERIVATIVES AS RHO-KINASE INHIBITORS 2017
  • Accetta, Alessandro
  • Rancati, Fabio
  • Capelli, Anna Maria
  • Clark, David Edward
  • Tisselli, Patrizia
  • Edwards, Christine
  • Bhalay, Gurdip
RU2778478C2
NEW AMIDE DERIVATIVE USED AS AN INHIBITOR OF DIALGLYCEROL O-ACYLTRANSFERASE 2 AND ITS USE 2020
  • Yoon, Seung Hyun
  • Joo, Hyun Woo
  • Seo, Bo Kyung
  • Lee, Eun Jin
  • Jung, Jin Young
  • Yoon, Su Young
  • Kwak, Young Shin
  • Cho, Woo Young
  • Jo, Min Mi
RU2810064C1
NEW INDOLIZINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM 2013
  • Le-Digare Terri
  • Kasara Patrik
  • Stark Zherom-Benua
  • Anlen Zhan-Mishel
  • Dejvidson Dzhejms Eduard Pol
  • Marri Dzhejms Bruk
  • Grem Kristofer Dzhon
  • Chen Itszen
  • Zhenes Olive
  • Khikman Dzhon
  • Depil Stefan
  • Le-Tiran Arno
  • Niergesh Miklosh
  • De-Nantej Gijom
RU2646223C2
NEW BIARYL DERIVATIVE USED AS INHIBITOR OF DIACYLGLYCEROL ACYLTRANSFERASE 2 AND ITS USE 2021
  • Yoon, Seung Hyun
  • Joo, Hyun Woo
  • Seo, Bo Kyung
  • Lee, Eun Jin
  • Jung, Jin Young
  • Yoon, Su Young
  • Cho, Woo Young
RU2808433C1
NEW PHENYLPYRIDINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE DERIVATIVE 2018
  • Kim, Wol-Young
  • Park, Jung-Eun
  • Bang, Keuk-Chan
  • Park, Joon-Seok
RU2748945C1
INHIBITOR COMPOUNDS 2013
  • Khelder Sven
  • Blagg Dzhulian
  • Solanki Savade
  • Vuduard Khannakh
  • Naud Sebasten
  • Bavetsias Vassilios
  • Sheldrejk Piter
  • Innochenti Paolo
  • Cheung Kvaj-Min Dz.
  • Atrash Betras
RU2673079C2

RU 2 705 577 C2

Authors

Bae In Hwan

Son Jung Beom

Han Sang Mi

Kwak Eun Joo

Kim Ho Seok

Song Ji Young

Byun Eun Young

Jun Seung Ah

Ahn Young Gil

Suh Kwee Hyun

Dates

2019-11-08Published

2012-12-27Filed