ANTICONVULSANT Russian patent published in 2019 - IPC A61K31/5377 A61P25/08 

Abstract RU 2705810 C1

FIELD: medicine; pharmacology.

SUBSTANCE: invention refers to medicine, particularly to pharmacology, and can be used to eliminate or prevent epileptic convulsions. Purpose of the invention is to search for new anticonvulsants among 7-oxycoumarin derivatives. Problem is solved using synthetic compound 7-(2-Morpholino-2-oxoethoxy)-2H-chromen-2-one.

EFFECT: in experiments on animals (mice) it is proved that the compound shows anticonvulsant activity, by 100 % protecting animals from death after LD50 nicotine introduction (14 mg/kg).

1 cl, 3 tbl

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RU 2 705 810 C1

Authors

Shabanov Petr Dmitrievich

Myznikov Leonid Vitalevich

Yakovleva Ekaterina Evgenevna

Makarov Valerij Gennadevich

Dates

2019-11-12Published

2018-12-28Filed