N-SUBSTITUTED (1S,4AR,5S)-METHYL-5-[2-(2'-OXO-2',5'-DIHYDRO1-H-PYRROL-3'-YL)ETHYL]-1,4A-DIMETHYL-6-METHYLENEDECAHYDRONAPHTHALENE-1-CARBOXYLATES HAVING ANTICONVULSANT ACTIVITY Russian patent published in 2010 - IPC C07D207/27 A61K31/4015 

Abstract RU 2385863 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a novel N-substituted (1S,4aR,5S)-methyl-5-[2-(2'-oxo-2',5'-dihydro-1H-pyrrol-3'-yl)ethyl]-1,4a-dimethyl-6-methylenedecahydronaphthalene-1-carboxylates of formula (I) having anticonvulsant activity. The compounds are obtained from plant material - needles or sap of Siberian cedar.

EFFECT: obtaining novel compounds with anticonvulsant activity.

2 tbl, 6 ex

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RU 2 385 863 C2

Authors

Shul'Ts Ehl'Vira Ehduardovna

Chernov Sergej Viktorovich

Tolstikova Tat'Jana Genrikhovna

Dolgikh Margarita Petrovna

Bolkunov Aleksej Viktorovich

Tolstikov Genrikh Aleksandrovich

Dates

2010-04-10Published

2008-04-21Filed