(1S,4a,5S,6R)-METHYL-5{2-[1-(2-AMINO-2-OXOETHYL)-2-OXOPYRROLIDIN-3-YL]ETHYL}-1,4a,6-TRIMETHYLDECAHYDRONAPHTHALENE-1-CARBOXYLATE, HAVING ANTICONVULSANT AND ANALGESIC ACTIVITY Russian patent published in 2010 - IPC C07D207/27 A61K31/4015 

Abstract RU 2385864 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a novel compound (1S,4aR,5S,6R)-methyl- 5{2-[1-(2-amino-2-oxoethyl)-2-oxopyrrolidin-2-yl]ethyl}-1,4a,6-trimethyldecahydronaphthalene-1-carboxylate of formula (I) , having anticonvulsant and analgesic activity. The compound is obtained from plant material - needles or sap of Siberian cedar.

EFFECT: obtaining a novel compound with anticonvulsant and analgesic activity.

3 tbl, 2 ex

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RU 2 385 864 C2

Authors

Chernov Sergej Viktorovich

Shul'Ts Ehl'Vira Ehduardovna

Tolstikova Tat'Jana Genrikhovna

Dolgikh Margarita Petrovna

Bolkunov Aleksej Viktorovich

Tolstikov Genrikh Aleksandrovich

Dates

2010-04-10Published

2008-04-21Filed