FUNCTIONALISED DERIVATIVES OF MORPHOLINYLANTHRACYCLINE Russian patent published in 2020 - IPC C07D498/14 A61K31/5383 A61K47/64 A61K47/68 A61P35/00 

Abstract RU 2715902 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to novel functionalized derivatives of morpholinylanthracycline, which have cytotoxic activity and are applicable for treating diseases such as cancer, cell proliferative diseases and viral infections. Also disclosed are pharmaceutical compositions containing said compounds, and methods of treating diseases using such compounds or pharmaceutical compositions containing them. Invention also relates to the use of these derivatives for producing conjugates.

EFFECT: functionalised derivatives of morpholinylanthracycline are proposed.

6 cl, 6 dwg, 1 tbl, 9 ex

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RU 2 715 902 C2

Authors

Lupi, Vittoria

Caruso, Michele

Beria, Italo

Dates

2020-03-04Published

2015-11-04Filed