POLYCYCLIC COMPOUND ACTING AS KINASE INHIBITOR Russian patent published in 2024 - IPC C07D471/04 C07D498/14 C07D519/00 A61K31/4375 A61K31/4985 A61K31/519 

Abstract RU 2826488 C1

FIELD: biotechnology; medicine.

SUBSTANCE: present invention relates to biotechnology and can be used in medicine. Invention discloses new non-peptide protein kinase inhibitors. Compounds according to the present invention are characterized by general formula (I) and represent a class of organic compounds containing tricyclic heteroaryl groups.

EFFECT: invention can be used in treating diseases in which there is an increased activity of CDK and/or TRK kinases.

18 cl, 27 ex, 2 tbl

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RU 2 826 488 C1

Authors

Zhang, Hancheng

Cheng, Xin

Jia, Wei

Cai, Congcong

Dates

2024-09-11Published

2021-01-11Filed