FIELD: pharmaceuticals.
SUBSTANCE: present invention relates to novel non-steroidal compounds which are effective modulators of the glucocorticoid receptor, and intermediate compounds for preparing them, to said compounds for use in therapy, pharmaceutical compositions containing said compounds, to methods of treating diseases with said compounds and use of said compounds in production of medicinal agents.
EFFECT: disclosed are nonsteroidal modulators of glucocorticoid receptors for local drug delivery.
12 cl, 4 tbl, 3 dwg, 81 ex
| Title |
Year |
Author |
Number |
| NITRILE-CONTAINING ANTIVIRAL COMPOUNDS |
2021 |
- Owen, Dafydd Rhys
- Pettersson, Martin Youngjin
- Reese, Matthew Richard
- Sammons, Matthew Forrest
- Tuttle, Jamison Bryce
- Verhoest, Patrick Robert
- Wei, Liuqing
- Yang, Xiaojing
- Yang, Qingyi
|
RU2786722C1 |
| NITRILE-CONTAINING ANTIVIRAL COMPOUNDS |
2021 |
- Ouen, Defidd Ris
- Pettersson, Martin Yungchin
- Riz, Mettyu Richard
- Semmons, Mettyu Forrest
- Tattl, Dzhejmison Brajs
- Verkhust, Patrik Robert
- Vej, Lyutsin
- Yan, Syaotszin
- Yan, Tsingyuj
|
RU2820150C2 |
| NEW AZABICYCLOHEXANE DERIVATIVES |
2023 |
- Belyi Petr Aleksandrovich
- Lopatukhin Eduard Iurevich
- Korolev Vladimir Lvovich
- Zaslavskaia Kira Iakovlevna
- Korliukov Aleksandr Aleksandrovich
- Buikin Petr Alekseevich
|
RU2811800C1 |
| COMPOUNDS TARGETING TAU PROTEIN AND RELATED USE THEREOF |
2017 |
- Crew, Andrew, P.
- Berlin, Michael
- Flanagan, John, J.
- Dong, Hanqing
- Ishchenko, Alexey
|
RU2805523C2 |
| AMIDES OF CONDENSED PIPERIDINE AS MODULATORS OF ION CHANNELS |
2014 |
- Deninno Majkl Pol
- Anderson Kori
- Konroj Erika Linn
- Friman Brajan A.
- Grotenkhejs Peter Diderik Yan
- Adida-Rua Sara Sabina
- Kharli Dennis Dzhejms
- Per Fabris Zhan Denis
- Silina Alina
- Yu Dzhonni
- Chzhou Tszinlan
|
RU2741810C2 |
| DIAMINE DERIVATIVES |
2003 |
- Okhta Tosikharu
- Komorija Satosi
- Josino Tosikharu
- Uoto Kouiti
- Nakamoto Jumi
- Naito Khirojuki
- Motizuki Akijosi
- Nagata Tsutomu
- Kanno Khidejuki
- Khaginoja Norijasu
- Josikava Kendzi
- Nagamoti Masatosi
- Kobajasi Siozo
- Ono Makoto
|
RU2333203C2 |
| GEMINALLY SUBSTITUTED CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS |
2014 |
- Chajlders Mettyu Llojd
- Fuller Piter
- Gerin Devid
- Katts Dzhejson Devid
- Pu Tsinlin
- Skott Mark E.
- Tompson Kristofer F.
- Martines Mishel
- Folkon Deniell
- Torres Luis
- Deng Jongki
- Kurukulasuriya Ravi
- Tszen Khunbo
- Baj Yunfyn
- Kun Norman
- Lyu Yujmej
- Chzhen Chzhisyan
|
RU2664533C2 |
| DERIVATIVES OF DIAMINES |
2002 |
- Okhta Tosikharu
- Komorija Satosi
- Josino Tosikharu
- Uoto Kouiti
- Nakamoto Jumi
- Naito Khirojuki
- Motizuki Akijosi
- Nagata Tsutomu
- Kanno Khidejuki
- Khaginoja Norijasu
- Josikava Kendzi
- Nagamoti Masatosi
- Kobajasi Suozo
- Ono Makoto
|
RU2319699C2 |
| SUBSTITUTED DIAMINOCARBOXAMIDE AND DIAMINOCARBONITRILE DERIVATIVES OF PYRIMIDINES, COMPOSITIONS THEREOF AND METHODS OF TREATING USE THEREOF |
2012 |
- Delgado, Mercedes
- Yoon, Won, Hyung
- Tikhe, Jayashree
- Satoh, Yoshitaka
- Romanow, William, J.
- Sloss, Marianne
- Paisner, David, A.
- Norris, Stephen
- Nagy, Mark, A.
- Moghaddam, Mehran, F.
- Mccarrick, Meg
- Lebrun, Laurie, Ann
- Hilgraf, Robert
- Erdman, Paul
- Elsner, Jan
- Bennett, Brydon, L.
|
RU2697712C2 |
| DIAMINE DERIVATIVES |
2002 |
- Okhta Tosikharu
- Komorija Satosi
- Josino Tosikharu
- Uoto Kouiti
- Nakamoto Jumi
- Naito Khirojuki
- Motizuki Akijosi
- Nagata Tsutomu
- Kanno Khidejuki
- Khaginoja Norijasu
- Josikava Kendzi
- Nagamoti Masatosi
- Kobajasi Siozo
- Ono Makoto
|
RU2314303C2 |
