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(19)

(11)

2 733 406

(13)

(51)

IPC

C07D213/71(2006-01-01)

C07D213/75(2006-01-01)

C07D241/18(2006-01-01)

A61K31/44(2006-01-01)

A61K31/4965(2006-01-01)

A61P29/00(2006-01-01)

A61P37/00(2006-01-01)

(21) (22)

Application

2017145928, 2016-06-03

(24)

Start date

2016-06-03

(22)

Actual filing date

2016-06-03

(45)

Published

2020-10-01

(72)

Inventor

Cals, Joseph Maria Gerardus BarbaraMachnik, DavidNabuurs, Sander BernardusSabuco, Jean-FrancoisSchio, Laurent

(73)

Holder

Lead Pharma Holding B.V.Sanofi

ROR GAMMA MODULATORS (RORΓ) Russian patent published in 2020 - IPC C07D213/71 C07D213/75 C07D241/18 A61K31/44 A61K31/4965 A61P29/00 A61P37/00

Abstract RU 2733406 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to novel compounds of formula I, as well as pharmaceutical compositions based thereon.

(formula I)

EFFECT: obtaining novel compounds suitable for treating RORγ-mediated diseases or conditions, such as rheumatoid arthritis, psoriasis, inflammatory bowel disease, Crohn's disease and multiple sclerosis.

12 cl, 39 ex

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RU 2 733 406 C2

Authors

Cals, Joseph Maria Gerardus Barbara

Machnik, David

Nabuurs, Sander Bernardus

Sabuco, Jean-Francois

Schio, Laurent

Dates

2020-10-01—Published

2016-06-03—Filed