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2 409 577

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IPC

C07D471/04(2006-01-01)

A61K31/551(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2007134226/04, 2006-02-14

(24)

Start date

2006-02-14

(22)

Actual filing date

2006-02-14

(45)

Published

2011-01-20

(72)

Inventor

Plate Ral'FZaman Gejdo Enni Rudol'FKhermkens Pedro Kharol'D KhanJans Khristian Gerardus Jokhannes MarijaBjuehjsman Rogir KhristianDe Man Adrianus Petrus AntoniusKonti Paolo Dzhovanni MartinoLasher Skott DzhejmsDokter Villem Khendrik Abrakham

(73)

Holder

N.V. Organon

GLUCOCORTICOID RECEPTOR NON-STEROID MODULATORS Russian patent published in 2011 - IPC C07D471/04 A61K31/551 A61P29/00

Abstract RU 2409577 C2

FIELD: chemistry.

SUBSTANCE: invention describes dibenzo[b,f]pyrido[1,2-d][1,4]diazepinyl derivatives of general formula I: or pharmaceutically acceptable salts thereof (values of radicals are listed in the claim), which are glucocorticoid receptor modulators.

EFFECT: derivatives can be used in treating immunological and inflammatory diseases.

11 cl, 49 ex

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RU 2 409 577 C2

Authors

Plate Ral'F

Zaman Gejdo Enni Rudol'F

Khermkens Pedro Kharol'D Khan

Jans Khristian Gerardus Jokhannes Marija

Bjuehjsman Rogir Khristian

De Man Adrianus Petrus Antonius

Konti Paolo Dzhovanni Martino

Lasher Skott Dzhejms

Dokter Villem Khendrik Abrakham

Dates

2011-01-20—Published

2006-02-14—Filed