FIELD: pharmaceuticals.
SUBSTANCE: invention refers to compounds presented by formulas (I)–(XVIII), or their pharmaceutically acceptable salts and pharmaceutical compositions based thereon.
EFFECT: there are prepared new compounds possessing PAR2 inhibitory activity suitable for treating inflammatory skin disease or inflammatory intestinal disease.
15 cl, 8 tbl, 24 ex
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| HETEROCYCLIC COMPOUND |
2018 |
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| DIAMINE DERIVATIVES |
2003 |
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| DERIVATIVES OF CYCLOHEXANE OR TETRAHYDROPYRANE OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS, OR HYDRATES, OR SOLVATES OF THESE COMPOUNDS, OR THEIR SALTS, INTERMEDIATE COMPOUNDS FOR THEIR SYNTHESIS AND FUNGICIDE AGENT |
1992 |
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RU2084439C1 |
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2019 |
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2016 |
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- Brooijmans Natasja
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2013 |
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RU2661896C2 |
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2000 |
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2021 |
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2014 |
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2002 |
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- Motizuki Akijosi
- Nagata Tsutomu
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