FUSED TRICYCLIC HETEROCYCLIC COMPOUNDS AS HIV INTEGRASE INHIBITORS Russian patent published in 2021 - IPC C07D471/16 A61K31/5025 A61P31/18 

Abstract RU 2740187 C2

FIELD: pharmaceuticals.

SUBSTANCE: present invention relates to fused tricyclic heterocyclic compounds of formula (I) and pharmaceutically acceptable salts thereof, pharmaceutical compositions based thereon and use for HIV integrase inhibition.

EFFECT: obtaining new compounds capable of inhibiting HIV integrase.

15 cl, 4 tbl, 35 ex

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RU 2 740 187 C2

Authors

Yu, Tao

Waddell, Sherman, T.

Graham, Thomas, H.

Zhang, Yonglian

Mccauley, John, A.

Stamford, Andrew, W.

Cai, Jiaqiang

Qi, Zhiqi

Dates

2021-01-12Published

2016-12-22Filed