N- (PHENYLSULPHONYL) BENZAMIDES AND RELATED COMPOUNDS AS BCL-2 INHIBITORS Russian patent published in 2021 - IPC C07D471/04 A61K31/437 A61P35/00 A61P35/02 

Abstract RU 2744358 C2

FIELD: organic chemistry.

SUBSTANCE: present invention relates namely to a compound or a pharmaceutically acceptable salt thereof selected from the group consisting of:

The invention also relates to a pharmaceutical composition and a method for treating cancer susceptible to inhibition of Bcl-2 proteins.

EFFECT: proposed new organic compounds, which are Bcl-2 protein inhibitors, suitable for cancer treatment.

9 cl, 4 dwg, 7 tbl, 20 ex

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RU 2 744 358 C2

Authors

Wang, Shaomeng

Chen, Jianyong

Dates

2021-03-05Published

2017-08-04Filed