PHARMACEUTICAL COMPOSITIONS CONTAINING WATER-INSOLUBLE ANTIPSYCHOTIC DRUG AND SORBITAN ESTERS Russian patent published in 2021 - IPC A61K9/10 A61K31/496 A61K31/381 A61K31/551 A61K47/14 A61K47/30 A61P25/18 

Abstract RU 2757859 C2

FIELD: medicine.

SUBSTANCE: present invention relates to the field of medicine, namely to a method for the treatment of central nervous system disorders, including the injection to a subject of therapeutically effective amount of a pharmaceutical composition containing (a) 20-30 weight percent of A-7 compound; (b) 0.2-1 weight percent of sorbitane laurate; (c) 0.05-0.8 weight percent of polysorbate 20, and (d) aqueous carrier; where the ratio of components (b) and (c) is from 5:1 to 1:1 by weight.

EFFECT: proposed is a method for the treatment of central nervous system disorders, which provides the injection of improved pharmaceutical composition containing sorbitane ester.

13 cl, 9 dwg, 4 tbl, 5 ex

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RU 2 757 859 C2

Authors

Vandiver, Jennifer

Remenar, Julius, F.

Deaver, Daniel, R.

Perry, Jason, M.

Hickey, Magali, B.

Dates

2021-10-21Published

2012-03-19Filed