Patenton — panteon of patents

(19)

RU

(11)

2 802 426

(13)

C2

(51)

IPC

C07D401/12(2006-01-01)

C07D401/14(2006-01-01)

C07D405/14(2006-01-01)

C07D413/14(2006-01-01)

C07D417/14(2006-01-01)

C07D471/04(2006-01-01)

A61K31/4439(2006-01-01)

A61K31/496(2006-01-01)

A61K31/4709(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2021121980, 2020-01-03

(24)

Start date

2020-01-03

(22)

Actual filing date

2020-01-03

(45)

Published

2023-08-28

(72)

Inventor

Bernales, SebastianPujala, BrahmamPanpatil, DayanandUreta Diaz, Gonzalo AndresBelmar, Sebastian

(73)

Holder

Praxis Biotech Llc

FIBROBLAST ACTIVATION PROTEIN INHIBITORS Russian patent published in 2023 - IPC C07D401/12 C07D401/14 C07D405/14 C07D413/14 C07D417/14 C07D471/04 A61K31/4439 A61K31/496 A61K31/4709 A61P35/00 

Abstract RU 2802426 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to a compound of formula (I), where R, L, X, Y, m are defined in the claims, and pharmaceutical compositions containing it, designed to modulate the fibroblast activation protein (FAP).

(I)

EFFECT: compounds and compositions can be used as medicinal products for the treatment of diseases or disorders mediated by fibroblast activation protein (FAP), including hyperproliferative diseases.

32 cl, 3 dwg, 6 tbl, 47 ex

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RU 2 802 426 C2

Authors

Bernales, Sebastian

Pujala, Brahmam

Panpatil, Dayanand

Ureta Diaz, Gonzalo Andres

Belmar, Sebastian

Dates

2023-08-28—Published

2020-01-03—Filed

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