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2 807 924

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IPC

C07J43/00(2006-01-01)

A61K31/58(2006-01-01)

A61P31/10(2006-01-01)

A61P31/12(2006-01-01)

(21) (22)

Application

2023106391, 2023-03-17

(24)

Start date

2023-03-17

(22)

Actual filing date

2023-03-17

(45)

Published

2023-11-21

(72)

Inventor

Sergeev Vladimir NikolaevichDavydova Nadezhda KonstantinovnaSadykova Vera SergeevnaSavinova Tatyana Stepanovna

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Institut Elementoorganicheskikh Soedinenij Im. A.N. Nesmeyanova Rossijskoj Akademii Nauk Ran)

N-SUBSTITUTED DERIVATIVES OF 6α-PIPERAZINOMETHYLANDROOST-4-EN-3,17-DIONE, HAVING ANTIMICROBIAL ACTIVITY, AND THEIR PRODUCTION METHOD Russian patent published in 2023 - IPC C07J43/00 A61K31/58 A61P31/10 A61P31/12

Abstract RU 2807924 C1

FIELD: chemistry; pharmaceuticals.

SUBSTANCE: group of inventions relates to compounds of N-substituted derivatives 6α-piperazinomethylandrost-4-ene-3,17-dione of general formula I, where R = CH₃, Ph, CH₂Pb, which has antibacterial and antifungal activity, as well as the method of their preparation.

EFFECT: group of inventions provides a compound with an antimicrobial effect and an effective method of its preparation.

9 cl, 1 tbl, 5 ex

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RU 2 807 924 C1

Authors

Sergeev Vladimir Nikolaevich

Davydova Nadezhda Konstantinovna

Sadykova Vera Sergeevna

Savinova Tatyana Stepanovna

Dates

2023-11-21—Published

2023-03-17—Filed