COMPOUND WITH ANTI-CANCER ACTIVITY Russian patent published in 2023 - IPC C07D215/44 C07D401/12 C07D401/14 C07D405/14 C07D409/14 C07D413/12 C07D413/14 C07D487/04 C07D487/08 C07D495/14 C07D519/00 A61K31/4985 A61K31/4704 A61K31/551 A61P35/00 

Abstract RU 2809763 C2

FIELD: chemistry; pharmaceuticals.

SUBSTANCE: invention relates to a compound of formula (I) or a pharmaceutically acceptable salt thereof, which has anticancer activity. The following is disclosed: a compound of formula (I) or a pharmaceutically acceptable salt thereof, as well as a pharmaceutical composition, drug and therapeutic agent based thereon for the treatment of diffuse large B-cell lymphoma (DLBCL). The use of the invention makes it possible to effectively treat diffuse large B-cell lymphoma (DLBCL). In the general formula (I), L1 and L2 are either the same or different and each represents a group represented by one formula selected from the group consisting of formulas (A) to (F), and S represents a group represented by one formula, selected from the group consisting of formulas (S1)–(S18).

EFFECT: obtaining a compound with anti-cancer activity.

20 cl, 18 tbl, 15 ex

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Authors

Uchida Kenji

Kawai Ryohei

Yamamoto Keisuke

Kanai Toshimi

Ikota Hideo

Imaeda Takashi

Yoshida Kei

Dates

2023-12-18Published

2019-03-29Filed