IMIDAZOPYRIDINE DERIVATIVE AND PHARMACEUTICAL PREPARATION CONTAINING IT AS AN ACTIVE INGREDIENT Russian patent published in 2024 - IPC C07D471/04 A61K31/437 A61K31/5377 A61K31/496 A61P35/00 A61P25/28 A61P1/16 A61P31/16

Abstract RU 2810973 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to imidazopyridine derivatives specified in claim 1 of the formula, which inhibit the action of a protein kinase, which is at least one enzyme selected from MLK1, MLK2, and MLK3. The invention also relates to pharmaceutical preparations containing these derivatives as an active ingredient.

EFFECT: obtaining new compounds and a pharmaceutical preparation based on them which can be used in medicine for the prevention or treatment of cancer, neurodegenerative disease, non-alcoholic steatohepatitis and influenza.

9 cl, 16 dwg, 11 tbl, 98 ex

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RU 2 810 973 C2

Authors

Lee, Jae Won

Son, Do Hyun

Kang, Nam Sook

Choi, Sung Wook

Dates

2024-01-09—Published

2020-08-31—Filed