NOVEL AMINOALKANOIC ACID DERIVATIVE CONTAINING BIPHENYL GROUP, AND ANTIFUNGAL PHARMACEUTICAL COMPOSITION CONTAINING IT Russian patent published in 2024 - IPC C07C237/20 A61K31/165 A61P31/10 

Abstract RU 2826219 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound of formula 1, where R1-R3, n and m are defined in the claim, a stereoisomer or a pharmaceutically acceptable salt thereof. Compound according to the invention exhibits excellent antifungal and fungicidal effects.

EFFECT: compound according to the invention exhibits a synergistic effect when used in combination with a common antifungal agent, has a wide spectrum of antifungal activity against a large number of fungal pathogens and can be widely used in fields, where it is necessary to use antifungal or fungicidal agents against human pathogenic fungi and animal pathogenic fungi, as well as phytopathogenic fungi.

19 cl, 3 dwg, 9 tbl, 94 ex

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RU 2 826 219 C2

Authors

Park, Ki Duk

Park, Jong Hyun

Kim, Hyeon Ji

Lee, Ye Rim

Kim, Siwon

Choi, Ji Won

Yeon, Seul Ki

Lee, Jong-Seung

Bahn, Yong-Sun

Cheong, Eunji

Lee, Kyung-Tae

Hong, Joohyeon

Dates

2024-09-05Published

2020-06-25Filed