COMPOSITIONS AND METHODS FOR TREATING METABOLIC AND HEPATIC DISORDERS Russian patent published in 2025 - IPC C07K14/605 A61K38/26 A61K47/54 A61P1/16 A61P13/12 

Abstract RU 2833318 C1

FIELD: medicine; pharmaceutics.

SUBSTANCE: invention relates to a double GIP/GLP-1 receptor agonist, which is a compound of formula I or a pharmaceutically acceptable salt thereof, where R1 is selected from a group consisting of -C(=O)(OZ1) and -P(=O)(X)(Y); R2 is selected from a group consisting of -C(=O)(OZ2) and -P(=O)(X)(Y); X and Y each represent -OR4; where R4, Z1 and Z2 are defined in the claims. Also disclosed is a pharmaceutical composition containing a compound of formula I, and a method of treating metabolic disorders and fatty liver diseases.

EFFECT: compositions and methods for treating metabolic and hepatic disorders are disclosed.

36 cl, 6 tbl, 10 ex

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RU 2 833 318 C1

Authors

Lian, Brajan

Barker, Dzheffri I.

Yagiz, Kader

Barns, Morin

Stivens, Erland

Dates

2025-01-17Published

2022-01-18Filed