FIELD: medicine; pharmaceutics.
SUBSTANCE: invention relates to a double GIP/GLP-1 receptor agonist, which is a compound of formula I or a pharmaceutically acceptable salt thereof, where R1 is selected from a group consisting of -C(=O)(OZ1) and -P(=O)(X)(Y); R2 is selected from a group consisting of -C(=O)(OZ2) and -P(=O)(X)(Y); X and Y each represent -OR4; where R4, Z1 and Z2 are defined in the claims. Also disclosed is a pharmaceutical composition containing a compound of formula I, and a method of treating metabolic disorders and fatty liver diseases.
EFFECT: compositions and methods for treating metabolic and hepatic disorders are disclosed.
36 cl, 6 tbl, 10 ex
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Authors
Dates
2025-01-17—Published
2022-01-18—Filed