CONJUGATED DRUG BASED ON TRICYCLIC POLYPEPTIDE AND ITS USE Russian patent published in 2025 - IPC A61K47/64 C07K7/08 C07K7/56 A61P35/00 

Abstract RU 2837445 C2

FIELD: chemistry; pharmaceutics.

SUBSTANCE: invention relates to a conjugated drug based on a tricyclic polypeptide, particularly a compound of formula (III), or a pharmaceutically acceptable salt thereof, and use thereof in treating solid tumours in which nectin-4 is overexpressed.

EFFECT: what is presented is a conjugated drug based on a tricyclic polypeptide for treating solid tumours in which nectin-4 is overexpressed.

10 cl, 4 dwg, 16 tbl, 9 ex

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RU 2 837 445 C2

Authors

Li, Huining

Xia, Jianhua

Jiang, Zhigan

He, Haiying

Chen, Shuhui

Dates

2025-03-31Published

2022-09-23Filed