HOMODETIC CYCLIC PEPTIDES SPECIFICALLY ACTING ON α4β7 INTEGRIN Russian patent published in 2022 - IPC C07K7/64 C07K7/54 A61K38/12 A61P29/00 A61P37/06 

Abstract RU 2773443 C2

FIELD: medicine.

SUBSTANCE: invention relates to α4β7 integrin antagonist, which is dimer containing two compounds of the formula (I), covalently bound to each other, its pharmaceutical composition and a method for the treatment of a condition related to biological α4β7 integrin function.

EFFECT: obtaining α4β7 integrin antagonist.

22 cl, 9 dwg, 3 tbl, 1 ex

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RU 2 773 443 C2

Authors

Vaskes, Manuel, Peres

Morshed, Montsur, M.

Kafal, Adam, Pol

Khiki, Dzhennifer, L.

Rafton, Endryu

Dates

2022-06-03Published

2018-05-10Filed