MONTELUKAST SALTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEREOF Russian patent published in 2025 - IPC C07D215/18 A61K31/137 A61K31/167 A61K31/47 A61P11/00 A61P11/06 A61P11/08 

Abstract RU 2840778 C2

FIELD: chemistry; pharmaceutics.

SUBSTANCE: invention relates to a salt of montelukast with β2 adrenergic agonist, where β2 adrenergic agonist is selected from formoterol and salbutamol. Method for preparing said montelukast salt, a pharmaceutical composition containing said montelukast salt and use of said montelukast salt as a medicinal agent are also provided.

EFFECT: obtaining novel montelukast salts having a synergistic therapeutic effect in treating allergen-caused respiratory tract dysfunctions.

14 cl, 18 dwg, 6 ex

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RU 2 840 778 C2

Authors

Caliendo, Giuseppe

Cirino, Giuseppe

Fiorino, Ferdinando

Frecentese, Francesco

Muscara', Marcelo, Nicolas

Perissutti, Elisa

Petti, Antonio

Roviezzo, Fiorentina

Santagada, Vincenzo

Severino, Beatrice

Dates

2025-05-28Published

2020-06-05Filed