PROCESS FOR PREPARING 3-QUINUCLIDINYL PROPIONIC ACID ESTERS Russian patent published in 1994 - IPC

Abstract RU 2005721 C1

FIELD: medicine. SUBSTANCE: products- 3-quinuclidinyl propionic acid esters of formula 1, wherein X- phenyl, fluorosubstituted phenyl or thienyl, Y- 5-member nitrogen-containing heterocycle selected from group consisting of imidazolyl, pyrazolyl, triazolyl or tetrazolyl, or their hydrochlorides. Reagent 1: compound of formula 2, wherein X and Y is as defined above. Reagent 2: lithium diisopropylamide or sodium hydride. Reagent 3: formaldehyde. Reaction conditions : reaction is carried our in organic solvent under cooling. EFFECT: increased production efficiency. 3 tbl

Similar patents RU2005721C1

Title Year Author Number
QUINUCLIDINE ESTERS, INTERMEDIATE COMPOUNDS FOR ITS SYNTHESIS, PHARMACEUTICAL COMPOSITION AND A METHOD OF TREATMENT 1992
  • Piter Ehdvard Kross
  • Alan Stobi
RU2117669C1
INDOLE DERIVATIVES OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS 1993
  • Dzhon I.Mehjkor[Us]
  • Martin Dzh.Uits[Gb]
RU2101283C1
INDOLE DERIVATIVES, SUBSTITUTED INDOLES, AND METHOD OF INHIBITING SEROTONIN 5HT RECEPTOR 1992
  • Dzhon I.Mehkor
RU2126399C1
SUBSTITUTED PYRAZOLES, PHARMACEUTICAL COMPOSITION BASED ON SAID, METHOD OF PATIENT TREATMENT, INTERMEDIATE COMPOUND 1993
  • Dzhen M.Brajt
  • Uillard M.Uehlch
RU2130453C1
AMINOSUBSTITUTED PYRAZOLES AND INTERMEDIATE AMINO SUBSTITUTED PYRAZINES 1993
  • Dzhen Majkl Brajt
RU2142455C1
METHOD OF SYNTHESIS OF TRIAZOLE DERIVATIVES 1991
  • Stefen Dzhejms Rehj[Gb]
  • Kennet Richardson[Gb]
RU2036194C1
PYRAZOLOPYRIMIDINES AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS 1993
  • Jukhping Liang Chen
RU2124016C1
COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA-2-ADRENERGIC RECEPTOR AGONIST ACTIVITY 2013
  • Rancati Fabio
  • Linney Ian
  • Knight Chris
  • Schmidt Wolfgang
RU2661877C2
1,2,4-TRIAZOLE DERIVATIVES OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS, PHARMACEUTICAL COMPOSITION AND INTERMEDIATE COMPOUNDS 1992
  • Rodzher Piter Dikinson[Gb]
  • Kennet Richardson[Gb]
RU2095358C1
INDOLE DERIVATIVES, THEIR OPTICAL ISOMERS AND PHARMACEUTICALLY ACCEPTABLE SALTS 1991
  • Dzhon Judzhin Makor[Us]
  • Martin Dzhejms Vites[Gb]
RU2095360C1

RU 2 005 721 C1

Authors

Piter Ehdvard Kross[Gb]

Alan Stoubi[Gb]

Dates

1994-01-15Published

1990-10-18Filed