AMINOSUBSTITUTED PYRAZOLES AND INTERMEDIATE AMINO SUBSTITUTED PYRAZINES Russian patent published in 1999 - IPC

Abstract RU 2142455 C1

FIELD: medicine. SUBSTANCE: described are new aminosubstituted pyrazoles of general formula: wherein R1-R3, A, Z and Y are as defined in claim 1. Said pyrazoles have antagonistic activity with respect to releasing factor of corticotropin. They are effective in treating wide range of diseases including stress induced disease. Also described are intermediate aminosubstituted pyrazines. EFFECT: improved properties of the title compounds. 13 cl, 36 ex, 4 tbl

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RU 2 142 455 C1

Authors

Dzhen Majkl Brajt

Dates

1999-12-10Published

1993-11-12Filed