FIELD: organic chemistry. SUBSTANCE: derivatives of imidazo(1,2-b) benzothiazoles of formula (I), , where R1 - cyclopropyl; R2 and R3 taken together mean group of formula II, , and formula III, , where X1 and X2 are similar or different, and every means hydrogen atom, C1-C5-alkyl, arylalkoxy, linear or branched C1-C5-alkoxy, or X1 and X2 taken together mean methylenedioxy-group. Synthesized compounds are used as antagonists of benzodiazepines. EFFECT: improved method of synthesis. 2 tbl
Title |
Year |
Author |
Number |
IMIDAZOBENZODIAZEPINES OR THEIR ADDITIVE SALTS WITH ACIDS |
1992 |
- Kolin Robert Gardner[Gb]
- Charl'Z Dzhon Robert Khedzhkok[Gb]
|
RU2041225C1 |
DERIVATIVES OF 3-CYCLOALKYLPROPENE-2-AMIDE OR THEIR ADDITIVE SALTS WITH MINERAL OR ORGANIC BASES, METHOD OF THEIR SYNTHESIS AND PHARMACEUTICAL COMPOSITION SHOWING ANTIINFLAMMATORY ACTIVITY |
1992 |
|
RU2072987C1 |
3-CYCLOALKYLPROPANEAMIDES SHOWING ANTIINFLAMMATORY AND IMMUNOSUPPRESSING ACTIVITY, METHOD OF THEIR SYNTHESIS, CYANAMIDE AND PHARMACEUTICAL COMPOSITION |
1991 |
- Filip Tomas Khambleton[Gb]
- Charl'Z Dzhon Robert Khedzhekok[Gb]
- Devid Pol Kej[Gb]
- Ehlizabet Ann Kuo[Gb]
- Vil'Fred Rodzher Tulli[Gb]
|
RU2073667C1 |
DERIVATIVES OF DIENE AMIDES, METHOD FOR THEIR PRODUCTION, INSECT ACARICIDE COMPOSITION AND METHOD FOR CONTROL OF INSECTS |
1992 |
- Dzhon Ehdvard Robinson[Gb]
- Zhorzh Stjuar Kokkeril[Gb]
|
RU2078076C1 |
2-CYANO-3-HYDROXYPROPENEAMIDES, METHODS OF THEIR SYNTHESIS AND A PHARMACEUTICAL COMPOSITION BASED ON SAID |
1994 |
|
RU2126387C1 |
AMIDES OF UNSATURATED ACIDS AND INTERMEDIATE PRODUCTS FOR THEIR PRODUCTION |
1992 |
- Robert Dzhon Blehjd[Gb]
- Dzhordzh Stjuart Kokerill[Gb]
- Dzhon Ehdvard Robinson[Gb]
|
RU2072351C1 |
STEROIDS, A METHOD OF SYNTHESIS OF STEROIDS, A METHOD OF SYNTHESIS OF 16-METHYLENESTEROIDS, COMPOUNDS |
1992 |
- Zhan Buavehn[Fr]
- Kristin Shove[Fr]
- Samir Zard[Lb]
|
RU2099346C1 |
AMIDES OF UNSATURATED ACIDS OR THEIR MOLES, METHOD FOR THEIR PRODUCTION AND INSECTICIDE OR ACARICIDE COMPOSITION |
1991 |
- Robert Dzhon Blehjd[Gb]
- Dzhordzh Stjuart Kokerill[Gb]
|
RU2086539C1 |
DERIVATIVES OF -PHENYL ALKANE ACIDS WHICH POSSES ANTIGLYCOCORTICOID, ANTIANDROGEN PROPERTIES |
1992 |
- Martin Mogilevski[Fr]
- Ljus'En Nedelek[Fr]
- Fransua Nik[Fr]
- Daniel' Filiber[Fr]
|
RU2041236C1 |
METHOD OF PRODUCING DERIVATIVES OF PYRIMIDO(2,1-B)BENZTHIAZOL |
0 |
- David Alan Roulends
- Serup Singkh Macharu
- Piter Uilfred Khejrsajn
|
SU1544191A3 |