DERIVATIVES OF IMIDAZO(1,2-b)BENZOTHIAZOLE AS ANTAGONISTS OF BENZODIAZEPINES Russian patent published in 1994 - IPC

Abstract RU 2014334 C1

FIELD: organic chemistry. SUBSTANCE: derivatives of imidazo(1,2-b) benzothiazoles of formula (I), , where R1 - cyclopropyl; R2 and R3 taken together mean group of formula II, , and formula III, , where X1 and X2 are similar or different, and every means hydrogen atom, C1-C5-alkyl, arylalkoxy, linear or branched C1-C5-alkoxy, or X1 and X2 taken together mean methylenedioxy-group. Synthesized compounds are used as antagonists of benzodiazepines. EFFECT: improved method of synthesis. 2 tbl

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RU 2 014 334 C1

Authors

Charl'Z Dzhon Robert Khedzhkok[Gb]

Dehvid Pol Kehj[Gb]

Dates

1994-06-15Published

1992-01-14Filed