FIELD: organic chemistry. SUBSTANCE: product: heterocyclic compounds of the formula (I) where R1, X, Y and B have the corresponding meanings, or their pharmaceutically acceptable additive acid salts, or heterocyclic compound N-oxide, or additive acid salt. These compounds were used in pharmaceutical compositions at concentration 0.5-730 mg per a dose. Synthesized compounds were used in medicine as antagonists of specific 5-hydroxytryptamine (5-HT) receptors for treatment patients with neuropsychiatric disorders. EFFECT: improved method of synthesis.
Title |
Year |
Author |
Number |
METHOD FOR PREPARING DERIVATIVES OF 4-OXOQUINOLINE OR CHROMAN OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS |
1991 |
- Terens Dzhejms Uord[Gb]
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|
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(ENDO)-N-[[(8-METHYL-8-AZABICYCLO-[3;2;1]-OCTANE-3-YL)-AMINO]- -CARBONYL]-2-(CYCLOPROPYLMETHOXY)-BENZAMIDE OR ITS PHARMACEUTICALLY ACCEPTABLE SALTS |
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|
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- Mansell Khovard Langkhehm
|
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1992 |
|
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1992 |
|
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|
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PROCESS FOR PREPARING DERIVATIVES OF INDOLE OR THEIR SALTS |
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|
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METHOD FOR PRODUCING DERIVATIVES OF HEXAHYDROAZEPINE,OR PIPERIDINE,OR PYRROLIDINE (VERSIONS) |
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|
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- Kristofer Jan Brajtuell
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|
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