FIELD: organic chemistry. SUBSTANCE: product: 2,3,4,5,6,7-hexahydro-1-[4-[1-[4-(2-methoxyphenyl)piperazinyl]]-2-phenylbutyryl]-1H-azepine, m. p. is 175-178 C. Reagent 1: 2,3,4,5,6,7-hexahydro-1H-azepine. Reagent 2: compound of the formula (I) HTIA. Reaction condition: in organic solvent medium. Synthesized compound is used in medicine for receptor 5- binding. EFFECT: improved method of synthesis. 7 cl
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