2-MERCAPTOBENZIMIDAZOLE DERIVATIVES HAVING SELECTIVE ANXIOLYTIC ACTIVITY Russian patent published in 1996 - IPC

Abstract RU 2061686 C1

FIELD: medicine. SUBSTANCE: 2- mercaptobenzimidazole derivatives having selective anxiolytic activity of formula wherein n is 0.2 or 3; R is allyl, dialkylamino or monocyclic saturated amino residue which may contain additional heteroatom, R¹ and R² are H, lower alkyl, alkoxy, or pharmaceutically acceptable salts obtained by alkylation of 2- mercaptobenzimidazole with suitable alkylating agents in aqueous alcoholic medium in the presence of bases. Structure of the compound of formula: . EFFECT: improved properties of the title products. 16 tbl

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RU 2 061 686 C1

Authors

Seredenin S.B.

Blednov Ju.A.

Savel'Ev V.L.

Mozhaeva T.Ja.

Ragimov Kh.S.

Jarkova M.A.

Dates

1996-06-10—Published

1994-06-10—Filed