FIELD: organic chemistry. SUBSTANCE: product: diazepinone derivatives of the formula (I) where: X - group =CH or nitrogen atom if B means bivalent residue of the formula (a): l = 1, 2, 3; m = 1, 2; n = 1-4; R' - H or C1-C6-alkyl and others. Reagent 1: compound of the formula (II). Reagent 2: carboxylic acid. Pharmaceutical composition exhibiting antimuscarinic activity has one derivative of diazepinone of the formula (I) taken at effective amount and pharmaceutically acceptable carrier. EFFECT: improved method of synthesis. 4 cl, 2 tbl
Title | Year | Author | Number |
---|---|---|---|
DERIVATIVES OF DIAZEPINONE, MIXTURES OF THEIR ISOMERS AND THEIR SALTS | 1992 |
|
RU2017740C1 |
METHOD OF PREPARING BENZODIAZEPINONE DERIVATIVES OR THEIR SALTS | 0 |
|
SU797578A3 |
DERIVATIVES OF DIPYRIDO-DIAZEPINE AND THEIR HYDRATES SHOWING BIOLOGICAL ACTIVITY | 1992 |
|
RU2040527C1 |
METHOD OF PREPARING PYRIDOBENZODIAZEPINONES OR SALTS THEREOF | 0 |
|
SU578878A3 |
PROCESS FOR PREPARING DIAZEPINONE DERIVATIVES | 0 |
|
SU1103795A3 |
DERIVATIVES OF PYRIDINE, THEIR ENANTIOMERS, CIS- OR TRANS-ISOMERS AND THEIR SALTS AND PHARMACEUTICAL COMPOSITION | 1992 |
|
RU2119915C1 |
0 |
|
SU331554A1 | |
METHOD FOR PRODUCING DIBENZODIAZEPINONE DERIVATIVES OR ACID-ADDITIVE SALTS THEREOF | 0 |
|
SU1301314A3 |
DERIVATIVES OF PYRIDYL, MIXTURE OF THEIR ISOMERS, OR INDIVIDUAL ISOMERS, OR THEIR PHYSIOLOGICALLY TOLERATED ADDITIVE SALTS SHOWING BIOLOGICAL ACTIVITY | 1991 |
|
RU2028292C1 |
METHOD OF PREPARING PYRIDOBENZODIAZEPINONES OR THEIR SALTS | 0 |
|
SU786900A3 |
Authors
Dates
1997-06-20—Published
1992-04-10—Filed