2,3-DIHYDRO-1,4-BENZODIOXINE-5-YL-PYRERAZINE DERIVATIVES AND SALTS THEREOF Russian patent published in 1998 - IPC

Abstract RU 2118322 C1

FIELD: medicine, organic technology. SUBSTANCE: 2,3-dihydro-1,4-benzodioxine-5-yl-pyperazine derivatives have formula I wherein R1 is halogen, lower alkyl or alkoxyl, hydroxyl or cyan group, m=1 or 2, n=0 or 1. A is alkylene chain comprising 2-6 carbon atoms which may be substituted by one or two lowers alkyl groups or by one phenyl group. B is methylene, ethylene, carbonyl, sulfunyl, sulfonyl or sulfur. Proposed compounds or salts thereof posses 5-HT1A-antagonist activity. EFFECT: improved quality of product. 1 tbl

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RU 2 118 322 C1

Authors

Jan Khartog

Bartolomeus Jokhannes Van Sten

Jokhannes Mos

Zhak Skhipper

Dates

1998-08-27Published

1994-07-04Filed