NOVEL TETRAAMINES SHOWING SELECTIVE AFFINITY TO M-CHOLINE RECEPTORS Russian patent published in 1999 - IPC

Abstract RU 2133245 C1

FIELD: organic chemistry. SUBSTANCE: invention relates to the novel N, N'-bis-(6-arylmethylaminohexyl)-1,4- and -1,3-diaminomethylbenzenes or α,w-polymethylene- and -α,w-polyoxapolymethylenediamines hydrochlorides or oxalates of the general formula: ArCH2NH(CH2)6NHCH2BCH2NH(CH2)6NHCH2Ar•4X where Ar is C6H5, 2-CH3OC6H4; B is 1,4-C6H4, 1,3-C6H4, ; X is HCl, H2C2O412 showing the selective affinity to the M2-choline receptors. EFFECT: new compounds indicated above, selective affinity to receptors. 2 dwg, 2 tbl, 2 ex

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RU 2 133 245 C1

Authors

Bespalov A.Ja.

Gorchakova T.L.

Dolgo-Saburov V.B.

Zlobina V.I.

Kosmachev A.B.

Libman N.M.

Lychakov A.V.

Podosinovikova N.P.

Ramsh S.M.

Shelkovnikov S.A.

Dates

1999-07-20Published

1995-04-07Filed