THIOPYRIDINES USED FOR CONTROL OF HELICOBACTER BACTERIA Russian patent published in 1999 - IPC

Abstract RU 2142459 C1

FIELD: organic chemistry, antibacterial agents. SUBSTANCE: invention relates to thiopyridines of the formula (I) where R1, R2 - H; R3 - H, C1-4-alkyl, C1-4-alkyl, C1-4-alkylcarbonyl, C2-4-alkenyl-carbonyl, halogen-C1-4-alkylcarbonyl or alkylsulfonyl that are substituted with R4; R4 is carboxy-group, C1-4-alkoxycarbonyl or -N(R14)R15; R15 - H, C1-4-alkyl or alkoxy-group; R6 is CmH2m-R6a radical where R6a - furan, thiophene, pyrrol, oxazole, isoxazole, thiazole, isothiazole, imidazole, pyrazole, triazole, tetrazole, thiadiazole, oxadiazole that can be substituted with R8 and R9 (other values see in p. 1 of the invention claim). Compounds are effective with respect to Helicobacter bacteria. EFFECT: new compounds indicated above, an antibacterial activity. 8 cl, 1 tbl, 13 ex

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RU 2 142 459 C1

Authors

Bernkhard Kol'

Gerkhard Grundler

Jorg Zenn-Bil'Finger

Guido Khanauer

Vol'Fgang-Aleksander Zimon

Peter Tsimmermann

Vol'Fgang Opferkukh

Dates

1999-12-10Published

1995-06-09Filed