DIARYL-5,6-CONDENSED HETEROCYCLIC ACIDS, PHARMACEUTICAL COMPOSITION, AND METHOD OF PROTECTION FROM EFFECTS OF LEUKOTRIENES Russian patent published in 2000 - IPC

Abstract RU 2154065 C2

FIELD: medicine. SUBSTANCE: described are new diaryl-5,6-condensed heterocyclic acids of general formula I: wherein are as defined in claim 1 which are antagonists of effects of lenkotrienes. Compounds are useful as antiasthmatic, antiallergic, antiinflammatory and cytoprotective agents. They are also useful in treating spasms of cerebrum, nephrite, kidney glomeruluses, hepatitis, endotoxicosis, uvent and tearing away of allotransplantate. Also described is pharmaceutical composition and method of protection from effects of leukotrienes. EFFECT: improved properties of the title compounds. 12 cl, 123 ex

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RU 2 154 065 C2

Authors

Robert N.Jang

Mark Label'

Iv Leblan

Ji Bin Ksjang

Cheuk L.Lau

Klod Djufren

Iv Garo

Dates

2000-08-10Published

1993-12-15Filed