FIELD: medicine. SUBSTANCE: described are new diaryl-5,6-condensed heterocyclic acids of general formula I: wherein are as defined in claim 1 which are antagonists of effects of lenkotrienes. Compounds are useful as antiasthmatic, antiallergic, antiinflammatory and cytoprotective agents. They are also useful in treating spasms of cerebrum, nephrite, kidney glomeruluses, hepatitis, endotoxicosis, uvent and tearing away of allotransplantate. Also described is pharmaceutical composition and method of protection from effects of leukotrienes. EFFECT: improved properties of the title compounds. 12 cl, 123 ex
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