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2 155 759

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IPC

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Application

98105820/04, 1998-03-25

(24)

Start date

1998-03-25

(22)

Actual filing date

1998-03-25

(45)

Published

2000-09-10

(72)

Inventor

Libman N.M.Zatsepin Eh.P.Pashkevich B.P.

(73)

Holder

Institut Toksikologii

AMINOALCOHOLS OF ACETYLENE ORDER SHOWING EXPRESSED M-CHOLINO-LYTIC PROPERTY AND WEAKLY SUPPRESSING CENTRAL NERVOUS SYSTEM Russian patent published in 2000 - IPC

Abstract RU 2155759 C2

FIELD: organic chemistry, medicine. SUBSTANCE: invention relates to biologically active compounds showing selective inhibitory effect on M-cholinoreactive systems and weakly SUPPRESSING the central nervous system activity. Invention describes the novel compounds: substituted aminobutynol hydrochlorides of the general formula (Ib-IVb) where R is ; NR12

is . The above indicated aminoalcohols are active and have low toxicity of M-cholinolytics of central effect, their activity exceeds that the known the most effective preparations but their effect on central nervous system is weaker. EFFECT: new compounds indicated above, valuable medicinal properties. 3 tbl

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RU 2 155 759 C2

Authors

Libman N.M.

Zatsepin Eh.P.

Pashkevich B.P.

Dates

2000-09-10—Published

1998-03-25—Filed

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