COMPOUNDS ACTIVE IN NOVEL SITE ON RECEPTOR-REGULATING CALCIUM CHANNELS AND USED FOR TREATMENT OF NEUROLOGICAL DISTURBANCES AND DISEASES Russian patent published in 2003 - IPC

Abstract RU 2201224 C2

FIELD: medicine. SUBSTANCE: invention relates to method of screening the therapeutical useful compound eliciting active as non-competitive antagonist of receptor-regulated calcium channel. Proposed method ensures to detect novel compounds and enhance effectiveness of treatment due to reduction of numbers of by-side effects. Invention can be used as neuroprotective, anticonvulsant agents and tranquilizers. EFFECT: valuable medicinal properties of compounds. 18 cl, 2 tbl

Similar patents RU2201224C2

Title Year Author Number
ARYLALKYLAMINES, COMPOSITIONS, METHODS OF TREATMENT AND DIAGNOSIS, METHOD OF IDENTIFICATION OF COMPOUND 1992
  • Ehdvard F.Nemet
  • Brehdford K.Van Vejgenen
  • Manuel' F.Balandrin
RU2147574C1
COMPOUNDS SHOWING ACTIVITY WITH RESPECT TO CALCIUM RECEPTORS (VERSIONS), PHARMACEUTICAL COMPOSITION AND METHODS OF TREATMENT (VERSIONS) 1995
  • Van Vagenen Brehdford K.
  • Moe Skott T.
  • Balandrin Manuehl' F.
  • Delmar Ehrik G.
  • Nemet Ehdvard F.
RU2195446C2
COMPOUNDS BEING ACTIVE AT A NEW SITE UPON RECEPTOR-OPERATED CALCIUM CANALS APPLIED FOR TREATING NEUROLOGICAL DISORDERS 1996
  • Alan L. Mjuller
  • Skott T. Moeh
  • Manuehl F. Balandrin
  • Ehrik Dzh. Delmar
  • Bredford K. Vanvagenen
  • Linda D. Artman
  • Robert M. Barmor
  • Dehril L. Smit
RU2246300C2
PHARMACEUTICAL COMPOSITION SHOWING ACTIVITY WITH RESPECT TO CALCIUM RECEPTOR, METHOD OF PATIENT TREATMENT, METHOD OF ANALYSIS OF COMPOUND EXHIBITING EFFECT ON ACTIVITY OF INORGANIC ION RECEPTOR, RECEPTOR-ENCODING NUCLEIC ACID, CALCIUM RECEPTOR 1993
  • Ehdvard F.Nemet
  • Ehdvard M.Braun
  • Stiven K.Khebert
  • Brehdford K. Van Vejgenen
  • Manuel' F.Balandrin
  • Forrest Kh.Fuller
  • Ehrik G.Del Mar
RU2146132C1
MONOCYCLIC L-NUCLEOSIDES, THEIR ANALOGUES AND USING 1997
  • Ramasejmi Kandasejmi
  • Tehm Robert
  • Ehverett Devron
RU2188828C2
PURINE L-NUCLEOSIDES, THEIR ANALOGUES AND USING 1997
  • Uong Guehndzhaj
  • Tehm Robert
  • Ehverett Devron
RU2183639C2
POLYPEPTIDE DERIVATIVES, METHOD OF CALCIUM CHANNEL INHIBITION 1993
  • Din M.Nejson Ii
  • Duglas Fillips
  • Nikolas Sakkomano
  • Robert A.Volkmann
RU2120945C1
POLYPEPTIDE OR ITS PHARMACEUTICALLY ACCEPTABLE SALTS 1993
  • Duglas Fillips[Us]
  • Mehri E.Kelli[Us]
  • Nikolas A.Sakkomano[Us]
  • Robert A.Vol'Kmann[Us]
RU2104286C1
POLYPEPTIDE OR ITS PHARMACEUTICALLY ACCEPTABLE SALT (VARIANTS); METHOD TO SUPPRESS THE ACTION OF AMINO ACID NEUROMEDIATORS 1993
  • Din M.Nehjson Ii[Us]
  • Robert T.Rono[Us]
  • Nikolas Sakkomano[Us]
  • Robert A.Volkman[Us]
  • Stiven D.Khek[Us]
RU2106358C1
RETINOID COMPOUNDS (VARIANTS), COMPOSITION, METHOD FOR ASSAY OF RETINOID HORMONE ANTAGONISTS, METHOD OF TREATMENT AND INTERMEDIATE SUBSTANCES 1996
  • Klejn Ehlliott S.
  • Dzhonson Alan T.
  • Stehndiven Ehndrju M.
  • Biard Richard L.
  • Gillett Sehmjuel Dzh.
  • Duong Tien T.
  • Nehgpehl Sanil
  • Valigonda Vid'Jasagar
  • Teng Min
  • Chandraratna Roshanta A.
RU2203884C2

RU 2 201 224 C2

Authors

Mjuller Alan L.

Van Vagenen Brehdford S.

Delmar Ehrik G.

Balandrin Manuel' F.

Mo Skott T.

Artman Linda D.

Barmor Robert M.

Dates

2003-03-27Published

1994-10-26Filed